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Search Results for " rp 5264 hydrochloride "

5

Compounds

Cat No. Product Name Synonyms Targets
T17066 Umbralisib hydrochloride RP5264 hydrochloride,TGR-1202 hydrochloride PI3K
Umbralisib hydrochloride is a novel PI3Kδ inhibitor (IC50 and EC50 of 22.2 nM and 24.3 nM, respectively). Umbralisib hydrochloride is also active against CK1ε (EC50: 6.0 μM).
T72527 Umbralisib sulfate TGR-1202 sulfate ; RP-5264 sulfate,TGR-1202 sulfate,RP-5264 sulfate
Umbralisib (TGR-1202) sulfate, an orally active compound, serves as a potent, selective inhibitor targeting both PI3Kδ and casein kinase-1-ε (CK1ε), with EC50 values of 22.2 nM and 6.0 μM, respectively. It demonstrates u...
T13140 Umbralisib R-enantiomer TGR-1202 R-enantiomer,RP5264 R-enantiomer PI3K
Umbralisib R-enantiomer (RP5264 R-enantiomer) is a delta inhibitor of PI3K and a less active enantiomer of TGR-1202. The IC50 of Umbralisib R-enantiomers against δPI3 kinase is at least 20 times lower than that of the in...
T72465 Umbralisib tosylate RP5264 tosylate,TGR-1202 tosylate ; RP5264 tosylate,TGR-1202 tosylate
Umbralisib Tosylate (TGR-1202) is a potent, selectively dual inhibitor targeting PI3Kδ and casein kinase-1-ε (CK1ε), demonstrating oral activity. With EC50 values of 22.2 nM and 6.0 μM for PI3Kδ and CK1ε respectively, it...
T4976 Umbralisib TGR-1202,RP5264,TGR 1202,TGR1202 PI3K
Umbralisib (TGR 1202) is a PI3Kδ inhibitor.
TargetMol